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Stable expression of human 5α-reductase type II in COS1 cells due to chromosomal gene integration : a novel tool for inhibitor identificationREICHERT, Wolfgang; MICHEL, Armin; HARTMANN, Rolf W et al.Journal of steroid biochemistry and molecular biology. 2001, Vol 78, Num 3, pp 275-284, issn 0960-0760Article

Design and synthesis of 1,3,5-trisubstituted 1,2,4-triazoles as CYP enzyme inhibitorsAL-SOUD, Yaseen A; HEYDEL, Michael; HARTMANN, Rolf W et al.Tetrahedron letters. 2011, Vol 52, Num 48, issn 0040-4039, 6307, 6372-6375 [5 p.]Article

Evaluation of 4'-substituted bicyclic pyridones as non-steroidal inhibitors of steroid 5α-reductaseMCCARTHY, Anna R; HARTMANN, Rolf W; ABELL, Andrew D et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 13, pp 3603-3607, issn 0960-894X, 5 p.Article

Protein-dynamics of the putative HCV receptor CD81 large extracellular loopNEUGEBAUER, Alexander; KLEIN, Christian D. P; HARTMANN, Rolf W et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 7, pp 1765-1769, issn 0960-894X, 5 p.Article

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Influence of DNA Template Choice on Transcription and Inhibition of Escherichia coli RNA PolymeraseHAUPENTHAL, Joerg; HÜSECKEN, Kristina; NEGRI, Matthias et al.Antimicrobial agents and chemotherapy. 2012, Vol 56, Num 8, pp 4536-4539, issn 0066-4804, 4 p.Article

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Synthesis and evaluation of a dimer of 2-(4-pyridylmethyl)-1-indanone as a novel nonsteroidal aromatase inhibitorGUPTA, Ranju; DHARAM PAUL JINDAL; JIT, Birinder et al.Archiv der Pharmazie (Weinheim). 2004, Vol 337, Num 7, pp 398-401, issn 0365-6233, 4 p.Article

Preparation and pharmacological profile of 7-(α-azolylbenzyl)-1H-indoles and indolines as new aromatase inhibitorsMARCHAND, Pascal; LE BORGNE, Marc; PALZER, Martina et al.Bioorganic & medicinal chemistry letters (Print). 2003, Vol 13, Num 9, pp 1553-1555, issn 0960-894X, 3 p.Article

Development of a test system for inhibitors of human aldosterone synthase (CYP11B2): screening in fission yeast and evaluation of selectivity in V79 cellsEHMER, Peter B; BUREIK, Matthias; BERNHARDT, Rita et al.Journal of steroid biochemistry and molecular biology. 2002, Vol 81, Num 2, pp 173-179, issn 0960-0760Article

N-(Pyridin-3-yl)benzamides as selective inhibitors of human aldosterone synthase (CYP11B2)ZIMMER, Christina; HAFNER, Marieke; ZENDER, Michael et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 1, pp 186-190, issn 0960-894X, 5 p.Article

Synthesis of amidinohydrazones and evaluation of their inhibitory effect towards aldosterone synthase (CYP11B2) and the formation of selected steroidsVOETS, Marieke; MÜLLER-VIEIRA, Ursula; MARCHAIS-OBERWINKLER, Sandrine et al.Archiv der Pharmazie (Weinheim). 2004, Vol 337, Num 7, pp 411-416, issn 0365-6233, 6 p.Article

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